luciferase in 1 — TargetMol Chemicals

Search Result

Search Results for " luciferase in 1 "

Compounds

Cat No.	Product Name	Synonyms	Targets
T38310	Luciferase-IN-1		Reactive Oxygen Species , Antibacterial , Antifungal
	Luciferase-IN-1 is a luciferase inhibitor that can be used to study bacterial and fungal infections.		Reactive Oxygen Species , Antibacterial , Antifungal
T9943	Firefly luciferase-IN-1		Others
	Firefly luciferase-IN-1 is a 2-benzylidene tetrahydronaphthone derivative and can be used as a firefly luciferase inhibitor in kit.		Others
T78389	Coelenteramine 400a	Bisdeoxycoelenterazine,Coelenterazine 400a
	Coelenteramine 400a (Coelenterazine 400a), a Coelenterazine derivative, serves as a substrate for Renilla luciferase (RLuc), facilitating the emission of blue light at 395 nm [1] [2]. This compound alters the bioluminesc...
T13364	YAP/TAZ inhibitor-1		ROCK
	YAP/TAZ inhibitor-1 is an inhibitor of YAP/TAZ (IC50 of <0.100 μΜ in firefly luciferase assay).		ROCK
T29336	2-Bromo-1-decanal	Decanal-1-14C, 2-bromo-, (R)-,2-Bromo(1-14C)-1-decanal
	2-Bromo-1-decanal was synthesized as an affinity labeling probe for the aliphatic aldehyde site of Vibrio harveyi luciferase. In the presence of excess amounts of this probe, the inactivation of bacterial luciferase occu...
T69241	MEISi-1
	MEISi-1 is a novel MEIS inhibitor (MEISi), significantly inhibiting MEIS-luciferase reporters in vitro and inducing murine (LSKCD34low cells) and human (CD34+, CD133+, and ALDHhi cells) HSC self-renewal ex vivo.
T78413	ETZ	C3-CA-DTZ
	ETZ (C3-CA-DTZ) represents a promising luciferase substrate (prosubstrate) that, upon activation by nonspecific esterase in vivo, facilitates enhanced delivery of luciferin to the brain [1].
T78419	LucPpy-IN-1
	LucPpy-IN-1 (compound 9) is an inhibitor of ATP-dependent luciferase from Photinus pyralis (lucPpy), exhibiting an IC50 value of 4.0 μM. It is utilized in research to assess the druggability [1] of the target enzyme.
T38223	N-(1-(3,4-Dihydroxyphenyl)propan-2-yl)oleamide
	N-(1-(3,4-Dihydroxyphenyl)propan-2-yl)oleamide binds to the cannabinoid 1 (CB1) receptor with a Ki value of 365 nM in a radioligand binding assay using rat brain homogenate. It has an EC50 value of 698 nM for the peroxis...
T37092	20-HEPE
	20-HEPE is a metabolite of eicosapentaenoic acid that is formed via ω-oxidation of EPA by cytochrome P450 (CYP) ω-oxidases, including human CYP4F3B. It activates peroxisome proliferator-activated receptor α (PPARα) in CO...
T70138	AZ0108
	AZ0108 is an orally bioavailable, potent PARP1,2,6 inhibitor that potently inhibits centrosome clustering and is suitable for in vivo efficacy and tolerability studies. AZ0108 has been utilized as in vitro tools and in ...
T81342	PyCTZ hydrochloride	Pyridyl CTZ hydrochloride
	PyCTZ (Pyridyl CTZ) hydrochloride, a pyridyl Coelenterazine (CTZ) analog, serves as an ATP-independent substrate for LumiLuc luciferase, producing intense blue bioluminescence when used with luciferases. This compound is...
T72056	KYN-101
	KYN-101 is a potent, selective synthetic antagonist of aryl hydrocarbon receptor (AHR) with IC50 of 22 nM in human HepG2 DRE-luciferase reporter assay and 23 nM in murine Hepa1 Cyp-luc assay.KYN-101 reverses IDO/TDO-medi...
T35800	MD001
	MD001 is a dual agonist of peroxisome proliferator-activated receptor α (PPARα) and PPARγ.1 It binds to PPARα and PPARγ (Kds = 9.55 and 0.14 μM, respectively) but does not bind to PPARβ/δ at concentrations up to 500 μM. ...
T36574	GW841819X	GW841819X
	GW841819X is an analogue of (+)-JQ1 and a novel inhibitor of BET bromodomains. GW841819X was a single enantiomer but of undefined chirality at the 4-position of the benzodiazepine ring3. GW841819X and JQ1 were recently d...